Patent application number | Description | Published |
20090054459 | Substituted indoles - Substituted indoles of the formula (I) and physiologically acceptable derivatives and salts thereof, in which R | 02-26-2009 |
20090291963 | SUBSTITUTED INDOLES - Substituted indoles of the formula (I) and physiologically acceptable derivatives and salts thereof, in which R | 11-26-2009 |
20090306122 | SUBSTITUTED TETRAHYDROPYRROLOQUINOLINE DERIVATIVES AS KINASE MODULATORS, ESPECIALLY OF TYROSINE AND RAF KINASES - Compound of the formula (I), in which X, R | 12-10-2009 |
20100160356 | NOVEL CYCLOBUTYL COMPOUNDS AS KINASE INHIBITORS - The invention relates to compounds of the formula I, to the preparation and use thereof for the preparation of a medicament for the treatment of diseases, in particular tumours and/or diseases in the formation or course of which protein kinases are involved. | 06-24-2010 |
20110059982 | AZAINDOLE COMPOUNDS FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS - Azaindole derivative compounds are described. The compounds have an optionally substituted azaindole core linked to a carbocyclic ring having at least one nitrogen atom and further bound to an optionally substituted aryl ring. A process for preparing these compounds, compositions comprising them, and methods of using them to treat disorders of the central nervous system are described. | 03-10-2011 |
20110105505 | THIAZOLYL PIPERIDINE DERIVATIVES - Compounds of the formula (I), in which R | 05-05-2011 |
20110207732 | AZAINDOLE DERIVATIVES - Compounds of the formula (I), in which X | 08-25-2011 |
20110263561 | Novel pyrrolidone derivatives for use as MetAP-2 inhibitors - Compounds of the formula (I), in which R, X, Y, Z, R | 10-27-2011 |
20110281859 | NOVEL HETEROCYCLIC COMPOUNDS AS METAP-2 INHIBITORS - Compounds of the formula I, in which D, X, Y, Z, R and R | 11-17-2011 |
20120252759 | THIAZOLE DERIVATIVES FOR THE TREATMENT OF DISEASES SUCH AS CANCER - Compounds of the formula Ia and Ib, in which R | 10-04-2012 |
20130158005 | PYRIMIDINE DERIVATIVES AS FAK INHIBITORS - Compounds of the formula (I), in which R | 06-20-2013 |
20130231519 | 1H-Pyrrolo[2,3 b]pyridine derivatives - 1H-Pyrrolo[2,3-b]pyridine compounds are inhibitors of cell proliferation/cell vitality and can be employed for the treatment of tumours. | 09-05-2013 |
20130245355 | 3-HETARYL-SUBSTITUTED PYRROLO[2,3 B]PYRIDINE DERIVATIVES AS PDK1 INHIBITORS - Compounds of the formula I in which Q, R | 09-19-2013 |
20130296274 | PYRROLIDINONES AS METAP-2 INHIBITORS - Compounds of the formula I in which R | 11-07-2013 |
20140100221 | 1H-Pyrrolo[2,3-b]Pyridine Derivatives - 1H-Pyrrolo[2,3-b]pyridine compounds are inhibitors of cell proliferation/cell vitality and can be employed for the treatment of tumours. | 04-10-2014 |
20140187551 | 7-AZAINDOLE DERIVATIVES SUITABLE FOR TREATMENT OF CANCERS - Compounds of the formula (I) in which R | 07-03-2014 |
20140221366 | Substituted Azaheterocycles for the Treatment of Cancer - The invention provides novel substituted azaheterocyclic compounds according to Formula (I), their manufacture and use for the treatment of hyperproliferative diseases, such as cancer. | 08-07-2014 |
20140371215 | 1-H-Pyrrolo[2,3-b]Pyridine Derivatives - 1H-Pyrrolo[2,3-b]pyridine compounds are inhibitors of cell proliferation/cell vitality and can be employed for the treatment of tumours. | 12-18-2014 |
20150031670 | CYCLIC AMIDES AS METAP-2 INHIBITORS - Compounds of the formula (I), in which R | 01-29-2015 |