Top Inventors for class "Organic compounds -- part of the class 532-570 series" |
Rank | Inventor's name | Country | City/State | Last publication | # of patent apps in this class |
1 | Gary L. Cantrell | US | Troy, IL | Apr 09, 2015 / 20150099773 - PROCESS FOR THE PREPARATION OF QUATERNARY N-ALKYL MORPHINAN ALKALOID SALTS | 35 |
2 | David W. Berberich | US | St. Peters, MO | Nov 26, 2015 / 20150335638 - (+)-MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF | 23 |
3 | Christopher W. Grote | US | Webster Groves, MO | Nov 26, 2015 / 20150335638 - (+)-MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF | 22 |
4 | Norbert Lui | DE | Odenthal | Oct 13, 2016 / 20160297766 - FUNGICIDE PYRAZOLE CARBOXAMIDES DERIVATIVES | 22 |
5 | Frank W. Moser | US | Arnold, MO | Jun 06, 2013 / 20130144053 - Process for the Production of Seven-Membered Lactam Morphinans | 21 |
6 | Gregory T. Whiteker | US | Carmel, IN | Oct 21, 2021 / 20210323923 - PREPARATION OF HALOGEN ANALOGS OF PICLORAM | 19 |
7 | Tao Jiang | US | St. Louis, MO | May 10, 2012 / 20120116086 - Sinomenine Derivatives and Processes for their Synthesis | 18 |
8 | Peter X. Wang | US | Clarkson Valley, MO | May 10, 2012 / 20120116086 - Sinomenine Derivatives and Processes for their Synthesis | 16 |
9 | James M. Renga | US | Indianapolis, IN | Jul 09, 2015 / 20150191428 - FLUOROPICOLINOYL FLUORIDES AND PROCESSES FOR THEIR PREPARATION | 16 |
10 | Peter X. Wang | US | Creve Coeur, MO | May 21, 2015 / 20150141649 - PREPARATION OF NORMORPHINANS | 14 |
11 | Gary Roth | US | Midland, MI | Sep 12, 2019 / 20190276431 - 4-((6-(2-(2,4-DIFLUOROPHENYL)-1,1-DIFLUORO-2-HYDROXY-3-(5-MERCAPTO-1H-1,2,- 4-TRIAZOL-1-YL)PROPYL)PYRIDIN-3-YL)OXY)BENZONITRILE AND PROCESSES OF PREPARATION | 14 |
12 | Beth Lorsbach | US | Indianapolis, IN | Jan 06, 2022 / 20220000114 - SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS COMPRISING 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE FOR FUNGAL CONTROL (MSI) | 13 |
13 | Kim E. Arndt | US | Carmel, IN | Oct 08, 2015 / 20150284377 - PROCESSES TO PRODUCE CERTAIN 2-(PYRIDINE-3-YL)THIAZOLES | 13 |
14 | Peter X. Wang | US | Chesterfield, MO | May 06, 2010 / 20100113788 - Process for the Preparation of 6-Alpha-Hydroxy-N-Alkylated Opiates | 13 |
15 | Qiang Yang | US | Zionsville, IN | Sep 12, 2019 / 20190276431 - 4-((6-(2-(2,4-DIFLUOROPHENYL)-1,1-DIFLUORO-2-HYDROXY-3-(5-MERCAPTO-1H-1,2,- 4-TRIAZOL-1-YL)PROPYL)PYRIDIN-3-YL)OXY)BENZONITRILE AND PROCESSES OF PREPARATION | 13 |
16 | Yuanming Zhu | US | Carmel, IN | Jun 07, 2018 / 20180155324 - 2-(2,4-DIFLUOROPHENYL)-1,1-DIFLUORO-1-(5-SUBSTITUTED-PYRIDIN-2-YL)-3-(1H-T- ETRAZOL-1-YL)PROPAN-2-OLS AND PROCESSES FOR THEIR PREPARATION | 13 |
17 | Ronald Ross, Jr. | US | Zionsville, IN | Nov 17, 2016 / 20160332987 - PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS | 12 |
18 | Michael Rack | DE | Eppelheim | May 19, 2016 / 20160137615 - Process for Manufacturing 4-Propargylated Amino-Benzoxazinones | 11 |
19 | Kura Rathnakar Reddy | IN | Hyderabad | Nov 25, 2021 / 20210363158 - PROCESS FOR THE PREPARATION OF SODIUM (2R,5S,13AR)-7,9-DIOXO-10-((2,4,6-TRIFLUOROBENZYL)CARBAMOYL)-2,3,4,5,7,9,- 13,13A-OCTAHYDRO-2,5-METHANOPYRIDO[1',2':4,5]PYRAZINO[2,1-B] [1,3] OXAZEPIN-8-OLATE AND ITS POLYMORPHIC FORM | 11 |
20 | David E. Podhorez | US | Midland, MI | Jul 01, 2021 / 20210198262 - METHOD OF PREPARATION OF FLORASULAM | 11 |
21 | Dasari Muralidhara Reddy | IN | Hyderabad | Oct 15, 2015 / 20150291574 - NOVEL POLYMORPHS OF AZILSARTAN | 11 |
22 | Sergii Pazenok | DE | Solingen | Jul 01, 2021 / 20210198180 - PROCESS FOR PRODUCING SUBSTITUTED 4-AMINOINDANE DERIVATIVES FROM 2-(HYDROXYALKYL)-ANILINES | 11 |
23 | Tomas Hudlicky | CA | St. Catharines | Nov 26, 2015 / 20150336971 - PROCESS FOR THE PREPARATION OF MORPHINE ANALOGS VIA METAL CATALYZED N-DEMETHYLATION/FUNCTIONALIZATION AND INTRAMOLECULAR GROUP TRANSFER | 11 |
24 | Bandi Parthasaradhi Reddy | IN | Hyderabad | Mar 19, 2020 / 20200087342 - C-3 NOVEL TRITERPENONE WITH C-17 REVERSE AMIDE DERIVATIVES AS HIV INHIBITORS | 11 |
25 | Mohan Prasad | IN | Gurgaon | Jun 30, 2016 / 20160185760 - PROCESS FOR THE PREPARATION OF MALIC ACID SALT OF SUNITINIB | 11 |
26 | Jian Li | US | Phoenix, AZ | Aug 13, 2015 / 20150228914 - METAL COMPOUNDS, METHODS, AND USES THEREOF | 11 |
27 | Eric Turner | US | Phoenix, AZ | Nov 05, 2015 / 20150318500 - Synthesis of Four Coordinated Platinum Complexes and Their Applications in Light Emitting Devices Thereof | 10 |
28 | Subo Liao | US | Ballwin, MO | Dec 30, 2021 / 20210403505 - PEPTIDES FOR TREATMENT OF MEDICAL DISORDERS | 10 |
29 | Rapolu Raji Reddy | IN | Hyderabad | Aug 21, 2014 / 20140235859 - PROCESS FOR THE RESOLUTION OF OMEPRAZOLE | 10 |
30 | Bobby N. Trawick | US | Florissant, MO | Nov 26, 2015 / 20150335638 - (+)-MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF | 9 |
31 | Carl Deamicis | US | Indianapolis, IN | Jun 07, 2018 / 20180155324 - 2-(2,4-DIFLUOROPHENYL)-1,1-DIFLUORO-1-(5-SUBSTITUTED-PYRIDIN-2-YL)-3-(1H-T- ETRAZOL-1-YL)PROPAN-2-OLS AND PROCESSES FOR THEIR PREPARATION | 9 |
32 | Stefan Abrecht | CH | Duggingen | Sep 10, 2015 / 20150252039 - Process For The Preparation Of Pyrido[2,1-a] Isoquinoline Derivatives By Catalytic Asymmetric Hydrogenation Of An Enamine | 9 |
33 | Shiro Tsubokura | JP | Takaoka-Shi | Jul 10, 2014 / 20140194629 - NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND METHOD FOR PRODUCING SAME | 9 |
34 | Michael Keil | DE | Freinsheim | Apr 30, 2015 / 20150119572 - Process for Manufacturing Aryloxyacetamides | 8 |
35 | Scott P. West | US | Midland, MI | Oct 08, 2015 / 20150284377 - PROCESSES TO PRODUCE CERTAIN 2-(PYRIDINE-3-YL)THIAZOLES | 8 |
36 | Tao Jiang | US | Chesterfield, MO | May 07, 2015 / 20150126742 - PRODUCTION OF 6-HYDROXY MORPHINANS WITHOUT THE ISOLATION OF INTERMEDIATES | 8 |
37 | Jian Bao | US | Chesterfield, MO | Nov 03, 2011 / 20110269964 - N-Alkylation of Opiates | 8 |
38 | Stefan Hildbrand | CH | Moehlin | Nov 26, 2015 / 20150336951 - Process For The Preparation Of A DPP-IV Inhibitor | 8 |
39 | Jens-Dietmar Heinrich | DE | Burscheid | Dec 27, 2012 / 20120330027 - PROCESS FOR THE PREPARATION OF 5-SUBSTITUTED 1-ALKYLTETRAZOLES | 8 |
40 | Mahavir Singh Khanna | IN | New Delhi | Apr 23, 2015 / 20150112085 - PURE CRYSTALLINE FORM II OF L-MALIC ACID SALT OF SUNITINIB AND PROCESSES FOR ITS PREPARATION | 8 |
41 | Yu Zhang | US | Carmel, IN | Aug 18, 2022 / 20220259176 - MOLECULE HAVING PESTICIDAL UTILITY, AND COMPOSITIONS, AND PROCESSES, RELATED THERETO | 8 |
42 | Nikolai (mykola) Ignatyev | DE | Duisburg | May 12, 2016 / 20160130286 - METHOD FOR PRODUCING SALTS HAVING MONOFLUORO-TRICYANOBORATE ANIONS | 8 |
43 | Rajesh Kumar Thaper | IN | Jammu | Jun 30, 2016 / 20160185760 - PROCESS FOR THE PREPARATION OF MALIC ACID SALT OF SUNITINIB | 8 |
44 | Xudong Wei | US | Ridgefield, CT | May 28, 2015 / 20150148322 - NOVEL PIPERIDINO-DIHYDROTHIENOPYRIMIDINE SULFOXIDES AND THEIR USE FOR TREATING COPD AND ASTHMA | 8 |
45 | Jian Li | US | Tempe, AZ | Jul 28, 2022 / 20220238833 - ORGANIC LIGHT-EMITTING DIODES WITH FLUORESCENT AND PHOSPHORESCENT EMITTERS | 8 |
46 | Kaitlyn Gray | US | Freeland, MI | Nov 17, 2016 / 20160332987 - PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS | 8 |
47 | Kurt Brandstadt | US | Midland, MI | Aug 13, 2015 / 20150224490 - Hydrosilylation Catalysts Made With Terdentate Nitrogen Ligands And Compositions Containing The Catalysts | 7 |
48 | Gary A. Roth | US | Midland, MI | Dec 03, 2015 / 20150344597 - PRODUCTION OF SUBSTITUTED PHENYLENE DIBENZOATE INTERNAL ELECTRON DONOR AND PROCATALYST WITH SAME | 7 |
49 | Josef Jirman | CZ | Praha | Sep 15, 2011 / 20110224441 - METHOD FOR THE PREPARATION OF DABIGATRAN AND ITS INTERMEDIATES | 7 |
50 | Ming-Shin Tzou | US | Midland, MI | Aug 13, 2015 / 20150224490 - Hydrosilylation Catalysts Made With Terdentate Nitrogen Ligands And Compositions Containing The Catalysts | 7 |
51 | Simon Cook | US | Midland, MI | Nov 26, 2015 / 20150337190 - Metal Containing Condensation Reaction Catalysts, Methods for Preparing the Catalysts, and Compositions Containing the Catalysts | 7 |
52 | Joseck M. Muhuhi | US | Midland, MI | Apr 28, 2016 / 20160115135 - PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS | 7 |
53 | Douglas C. Bland | US | Midland, MI | Nov 19, 2015 / 20150329509 - PROCESSES FOR THE PREPARATION OF ENAMINES | 7 |
54 | Binh Nguyen | US | Midland, MI | Aug 13, 2015 / 20150224490 - Hydrosilylation Catalysts Made With Terdentate Nitrogen Ligands And Compositions Containing The Catalysts | 7 |
55 | Pius Waldmeier | CH | Wegenstetten | Mar 24, 2016 / 20160083378 - NOVEL PROCESSES FOR THE MANUFACTURE OF PROPANE-1-SULFONIC ACID (3-[5-(4-CHLORO-PHENYL)-1H-PYRROLO[2,3-b]PYRIDINE-3-CARBONYL]-2,4-DIFLUOR- O-PHENYL)-AMIDE | 7 |
56 | Bo Qu | US | Brookfield, CT | Jun 07, 2018 / 20180155377 - NOVEL CHIRAL DIHYDROBENZOAZAPHOSPHOLE LIGANDS AND SYNTHESIS THEREOF | 7 |
57 | Geoff G.z. Zhang | US | Libertyville, IL | Apr 19, 2018 / 20180105510 - SALT AND CRYSTALLINE FORMS THEREOF OF A DRUG | 7 |
58 | Avril Surgenor | BE | Waterloo | May 26, 2016 / 20160145395 - Telomerisation Of Cyclic Polyorganosiloxanes | 7 |
59 | Enos Kiremire | NA | Windhoek | Jun 20, 2013 / 20130158267 - METHOD OF SYNTHESIZING THE COMPLEX [ZN(NNS)2] ACTIVE AGAINST THE MALARIA PARASITE PLASMODIUM | 7 |
60 | Oded Arad | IL | Rehovot | Aug 04, 2011 / 20110185796 - CISATRACURIUM DERIVATIVES, PREPARATION AND USES THEREOF | 6 |
61 | Gary David Annis | US | Landenberg, PA | Jul 13, 2017 / 20170197925 - METHOD FOR PREPARING 3-TRIFLUOROMETHYL CHALCONES | 6 |
62 | Joseph P. Haar, Jr. | US | Edwardsville, IL | Apr 09, 2015 / 20150099773 - PROCESS FOR THE PREPARATION OF QUATERNARY N-ALKYL MORPHINAN ALKALOID SALTS | 6 |
63 | Kwee Hyun Suh | KR | Suwon-Si | Oct 22, 2015 / 20150299185 - NOVEL IMIDAZOPYRIDINE DERIVATIVES AS A TYROSINE KINASE INHIBITOR | 6 |
64 | Rajendra Narayanrao Kankan | IN | Mumbai | Dec 29, 2016 / 20160374999 - RIFAXIMIN | 6 |
65 | Zixing Wang | CN | Shanghai | Nov 05, 2015 / 20150318500 - Synthesis of Four Coordinated Platinum Complexes and Their Applications in Light Emitting Devices Thereof | 6 |
66 | Helge Alfred Reisch | US | Westerly, RI | Oct 17, 2019 / 20190314364 - ACETATE SALT OF BUPRENORPHINE AND METHODS FOR PREPARING BUPRENORPHINE | 6 |
67 | Helmut Reichelt | DE | Neustadt | Aug 13, 2015 / 20150225418 - CONVENIENTLY PREPARED NAPHTHALENE AND PERYLENE DERIVATIVES AS BUILDING BLOCKS FOR ORGANIC ELECTRONIC MATERIALS AND DYESTUFF | 6 |
68 | Karsten Koerber | DE | Eppelheim | Dec 27, 2018 / 20180368404 - 3-PYRIDYL HETEROBICYCLIC COMPOUND FOR CONTROLLING INVERTEBRATE PESTS | 6 |
69 | Eric Dowdy | US | Foster City, CA | Jan 07, 2016 / 20160002186 - METHODS AND INTERMEDIATES FOR PREPARING PHARMACEUTICAL AGENTS | 6 |
70 | Kaoru Noda | JP | Takaoka-Shi | Jun 05, 2014 / 20140155615 - COMPOUND CONTAINING PYRIDINE RING AND METHOD FOR PRODUCING HALOGENATED PICOLINE DERIVATIVE AND TETRAZOLYLOXIME DERIVATIVE | 6 |
71 | Catherine E. Thomasson | US | Webster Groves, MO | Nov 03, 2011 / 20110269964 - N-Alkylation of Opiates | 6 |
72 | Scott D. Larsen | US | South Lyon, MI | May 26, 2016 / 20160145251 - INHIBITORS OF MYOCARDIN-RELATED TRANSCRIPTION FACTOR AND SERUM RESPONSE FACTOR (MRTF/SRF)-MEDIATED GENE TRANSCRIPTION AND METHODS FOR USE OF THE SAME | 6 |
73 | Mathai Mammen | US | Menlo Park, CA | Sep 17, 2020 / 20200290966 - BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS | 6 |
74 | Ales Machara | CZ | Brevnov | Nov 26, 2015 / 20150336971 - PROCESS FOR THE PREPARATION OF MORPHINE ANALOGS VIA METAL CATALYZED N-DEMETHYLATION/FUNCTIONALIZATION AND INTRAMOLECULAR GROUP TRANSFER | 6 |
75 | Yasutaka Takada | JP | Funabashi-Shi | Jun 30, 2016 / 20160185734 - METHOD FOR PRODUCING OPTICALLY ACTIVE 5-HYDROXY-3-KETOESTER | 6 |
76 | Hiroki Inoue | JP | Takaoka-Shi | Nov 19, 2015 / 20150329472 - HALOGENATED ANILINE AND METHOD FOR PRODUCING SAME | 6 |
77 | Steven P. Tanis | US | Carlsbad, CA | Apr 19, 2018 / 20180105551 - TRINUCLEOTIDE MRNA CAP ANALOGS | 6 |
78 | Raymond Kwong | US | Plainsboro, NJ | Jun 22, 2017 / 20170179394 - ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES | 6 |
79 | David M. Barnes | US | Lake Villa, IL | Apr 19, 2018 / 20180105510 - SALT AND CRYSTALLINE FORMS THEREOF OF A DRUG | 6 |
80 | Shao Hong Zhou | US | Commack, NY | Jan 26, 2017 / 20170022160 - PROCESSES FOR PREPARING HETEROCYCLIC COMPOUNDS INCLUDING TRANS-7-OXO-6-(SULPHOOXY)-1,6-DIAZABICYCLO[3,2,1]OCTANE-2-CARBOXAMIDE AND SALTS THEREOF | 5 |
81 | Robert Send | DE | Karlsruhe | Aug 25, 2022 / 20220268635 - METHOD AND DEVICE FOR MONITORING RADIATION | 5 |
82 | Ingmar Bruder | DE | Mutterstadt | Jun 22, 2017 / 20170178823 - BORON CONTAINING PERYLENE MONOIMIDES, A PROCESS FOR THEIR PRODUCTION, THEIR USE AS BUILDING BLOCKS FOR THE PRODUCTION OF PERYLENE MONOIMIDE DERIVATIVES, MONOIMIDE DERIVATIVES AND THEIR USE IN DYE-SENSITIZED SOLAR CELLS | 5 |
83 | Gwan Sun Lee | KR | Seoul | Feb 25, 2016 / 20160051696 - POLYPEPTIDE COMPLEX COMPRISING NON-PEPTIDYL POLYMER HAVING THREE FUNCTIONAL ENDS | 5 |
84 | Michael James Rishel | US | Rensselaer, NY | Aug 25, 2011 / 20110206609 - FLUOROALKYL TETRABENAZINE CARBINOL COMPOUNDS AS IMAGING AGENTS AND PROBES | 5 |
85 | Ralph Diodone | DE | Breisach | Nov 26, 2015 / 20150336951 - Process For The Preparation Of A DPP-IV Inhibitor | 5 |
86 | Antonio Zanotti-Gerosa | GB | Cambridge | Mar 03, 2016 / 20160060217 - Processes | 5 |
87 | Robert E. Halvachs | US | Belleville, IL | Apr 09, 2015 / 20150099773 - PROCESS FOR THE PREPARATION OF QUATERNARY N-ALKYL MORPHINAN ALKALOID SALTS | 5 |
88 | Akira Nishiyama | JP | Takasago-Shi | Jun 30, 2022 / 20220204451 - METHOD FOR PRODUCING A VADADUSTAT INTERMEDIATE | 5 |
89 | Ikuo Kushida | JP | Tsukuba | Oct 21, 2021 / 20210323972 - CRYSTALS OF PYRANODIPYRIDINE COMPOUND | 5 |
90 | Brian C. Austad | US | Tewksbury, MA | Aug 04, 2022 / 20220242832 - PROCESS FOR PREPARING XPO1 INHIBITORS AND INTERMEDIATES FOR USE IN THE PREPARATION OF XPO1 INHIBITORS | 5 |
91 | Michael Cyr | US | League City, TX | Dec 24, 2015 / 20150368200 - METHOD FOR SYNTHESIZING PIRFENIDONE | 5 |
92 | Peter L. Johnson | US | Indianapolis, IN | Oct 02, 2014 / 20140296533 - PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-CHLORO-6-(SUBSTITUTED)PICOLINATES | 5 |
93 | József Barkóczy | HU | Budapest | Jun 05, 2014 / 20140155614 - PHARMACEUTICAL INTERMEDIATES AND PROCESS FOR THE PREPARATION THEREOF | 5 |
94 | Brian Orr | US | O'Fallon, MO | Mar 22, 2012 / 20120071659 - Process for the Preparation of Sufentanil Base and Related Compounds | 5 |
95 | James R. Zeller | US | Scottsdale, AZ | Dec 25, 2014 / 20140378687 - Synthesis for Thiazolidinedione Compounds | 5 |
96 | Balázs Volk | HU | Budapest | Mar 19, 2020 / 20200087269 - PROCESS FOR THE PRODUCTION OF OZANIMOD | 5 |
97 | Koichi Ito | JP | Tsukuba | May 22, 2014 / 20140142315 - METHOD FOR PRODUCING 1,2-DIHYDROPYRIDINE-2-ONE COMPOUND | 5 |
98 | Frank Xing Chen | US | Plainsboro, NJ | May 26, 2016 / 20160145256 - PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 8-[-METHYL]-8-PHENYL-1,7-DIAZA-SPIRO[4.5]DECAN-2-ONE COMPOUNDS | 5 |
99 | Ji Xie | US | Edison, NJ | May 26, 2016 / 20160145256 - PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 8-[-METHYL]-8-PHENYL-1,7-DIAZA-SPIRO[4.5]DECAN-2-ONE COMPOUNDS | 5 |
100 | Chava Satyanarayana | IN | Secunderabad | Jun 09, 2011 / 20110137039 - PROCESS FOR THE PREPARATION OF MONTELUKAST AND ITS SALTS | 5 |